Protein Import: The Cytotoxic Colicins
Hypothesesfor the pathway and mechanisms of import into E. coli of the cytotoxic E colicins are partly based on structures of a complex of the colicin with its outer membrane vitamin B12 receptor (BtuB), which the colicins parasitize for import. A 2.75 Å structure of the complex of the receptor-binding domain of the endoribonucleolytic colicin E3 showed the elongate 100 Å long colicin domain to be bound in an oblique mode, in which it appears to be ‘fishing,’ for a second outer membrane receptor-translocator (Nature Structural Biology , 10, 948-954, 2003). A similar structure has been obtained with the receptor binding domain of colicin E2 (Sharma et al., JBC, 2007). Circular dichroism and electrophysiological studies imply that the colicin is first bound tightly to the extracellular surface of BtuB, is unfolded upon binding, and then uses another very abundant outer membrane protein, OmpF, for translocation (Biochemistry, 45:10199-10207, 2006, . Biol. Chem, J. Biol. Chem. 2007. 282: 23163-23170). It is proposed that colicin import across the outer membrane involves formation of a ‘translocon’ between BtuB and OmpF. A 1.6 Å structure has recently been obtained for OmpF (Yamashita et al., in preparation, 2007). A structure of the BtuB vitamin B12 receptor has recently been obtained, in collaboration with M. Caffrey, by crystallization in the lipid cubic phase (Cherezov et al., 2006). At 1.95 Å resolution, it is the highest resolution structure of a membrane protein not related to bacteriorhodopsin to be obtained by the in meso approach to crystallization.
Alpha-Synuclein
α-Synuclein, a 140 amino acid cytosolic protein implicated in the pathogenesis of Parkinson's Disease (PD), can exert its cellular function through interaction with membranes. Studies that we have carried out with J. - C. Rochet showed that monomeric synuclein in an alpha-helical conformation can form specific ion channels in planar bilayer membranes (Zakharov et al., Biochemistry, 2007). These channels must result from the formation of a trans-membrane oligomer of defined structure. The synuclein channels could have a positive function in the metabolism of synaptic membranes.

